Selective Bibliography of Dr. Terrence Burke
Chemical Biology Laboratory, NCI

Wednesday, November 16, 2022

1.  Tsuji K, Hymel D, Ma B, Tamamura H, Nussinov R, Burke TR, Jr.
Development of ultra-high affinity bivalent ligands targeting the polo-like kinase 1
RSC Chemical Biology 3 (9):1111-1120 Aug 31 2022

2.  Zhao XZ, Kiselev E, Lountos GT, Wang W, Tropea JE, Needle D, Hilimire TA, Schneekloth JS, Jr., Waugh DS, Pommier Y, Burke TR, Jr.
Small molecule microarray identifies inhibitors of tyrosyl-DNA phosphodiesterase 1 that simultaneously access the catalytic pocket and two substrate binding sites
Chemical Science 12 (11):3876-3884 Jan 28 2021
  
3.  Smith SJ, Zhao XZ, Passos DO, Pye VE, Cherepanov P, Lyumkis D, Burke TR, Jr., Hughes SH
HIV-1 Integrase Inhibitors with Modifications That Affect Their Potencies against Drug Resistant Integrase Mutants
ACS Infectious Diseases 7 (6):1469-1482 Jun 11 2021
   
4.  Hymel D, Tsuji K, Grant RA, Chingle RM, Kunciw DL, Yaffe MB, Burke TR, Jr.
Design and synthesis of a new orthogonally protected glutamic acid analog and its use in the preparation of high affinity polo-like kinase 1 polo-box domain - binding peptide macrocycles
Organic & Biomolecular Chemistry 19 (36):7843-7854 Sep 22 2021

5.  Passos DO, Li M, Józwik IK, Zhao XZ, Santos-Martins D, Yang R, Smith SJ, Jeon Y, Forli S, Hughes SH, Burke TR, Jr., Craigie R, Lyumkis D
Structural basis for strand-transfer inhibitor binding to HIV intasomes
Science 367 (6479):810-814 Feb 14 2020

6.  Miller SE, Tsuji K, Abrams RPM, Burke TR, Jr., Schneider JP
Uncoupling the Folding-Function Paradigm of Lytic Peptides to Deliver Impermeable Inhibitors of Intracellular Protein-Protein Interactions
Journal of the American Chemical Society 142 (47):19950-19955 Nov 25 2020
 
7.  Zhao XZ, Smith SJ, Maskell DP, Métifiot M, Pye VE, Fesen K, Marchand C, Pommier Y, Cherepanov P, Hughes SH, Burke TR, Jr.
Structure-Guided Optimization of HIV Integrase Strand Transfer Inhibitors
Journal of Medicinal Chemistry 60 (17):7315-7332 Sep 14 2017

8.  Zhao XZ, Smith SJ, Maskell DP, Metifiot M, Pye VE, Fesen K, Marchand C, Pommier Y, Cherepanov P, Hughes SH, Burke TR, Jr.
HIV-1 Integrase Strand Transfer Inhibitors with Reduced Susceptibility to Drug Resistant Mutant Integrases
ACS Chemical Biology 11 (4):1074-81 Apr 15 2016
 
9.  Zhao XZ, Smith SJ, Métifiot M, Marchand C, Boyer PL, Pommier Y, Hughes SH, Burke TR, Jr.
4-amino-1-hydroxy-2-oxo-1,8-naphthyridine-containing compounds having high potency against raltegravir-resistant integrase mutants of HIV-1
Journal of Medicinal Chemistry 57 (12):5190-202 Jun 26 2014

10.  Liu F, Park JE, Qian WJ, Lim D, Gräber M, Berg T, Yaffe MB, Lee KS, Burke TR, Jr.
Serendipitous alkylation of a Plk1 ligand uncovers a new binding channel
Nature Chemical Biology 7 (9):595-601 Jul 17 2011